噻啶

5 H-Thiazolo [3,2-a] pyrimidine derivatives were found to be active acetylcholinesterase inhibitors.

5H-噻唑并[3，2-a]嘧啶类化合物是潜在的乙酰胆碱酯酶抑制剂。

The center can finish various kinds of reactions, such as reactions in low temperature（-80℃）and high temperature（300℃）, hydrogenation reactions and so on. Especially in synthesizing primidine, pyridine, thiophene, quinoline and boronic acid, Yield lies at the leading level in China.

研发中心可以按客户需求完成各种低温（-80℃）、高温（300℃）、高压氢化等反应，尤其在嘧啶、吡啶、喹啉、噻吩及有机硼酸类化合物的合成方面，博鸿在国内同行业中处于领先水平。

Further aza-Wittig reactions of iminophosphorane 3 with aromatic isocyanates gave the carbodiimide s 4, which were reacted with secondary amines to give 2-dialkylamino-thieno[2,3-d]pyrimidin-4(3H)-ones 6 in the presence of catalytic amounts of EtO-Na+ in 58%～82%.

应用膦亚胺3与芳基异氰酸酯的氮杂Wittig反应，生成的碳二亚胺4，再与仲胺作用得到中间体5，而后在醇钠的催化下关环制得2-二烷氨基噻吩并[2，3-d]嘧啶-4(3H)-酮衍生物6，产率为58%～82

Three series of donor-acceptorπ-conjugated molecules 1, 2, and 3 have been designed and synthesized with a N, N-dimethylamino, Julolidine group (2,3,6,7-tetrahydro-1H, 5H-pyrido[3, 2, 1-ij]quinolinyl), or N, N-diphenylamino group as the donor moiety, a phenylvinyl or thienylvinyl unit as the bridge, and a bromide or aldehyde group as the acceptor moiety.

本文设计并合成了1、2、3三个系列的D-π-A型化合物(Donor-Acceptorπ-conjugated compounds)，在化合物分子中引入久洛尼啶基团(2，3，6，7-tetrahydro-1H，5H-pyrido-[3，2，1-ij]quinolinyl)，N，N-二甲基氨基，或N，N-二苯基氨基为供电子基团，以苯乙烯基或噻吩乙烯基为桥链，以溴原子或醛基为吸电子基团。

METHODS: A randomized controlled study was carried out to compare the efficacy of a single dose of 3 or 2 tablets of albendazole composite versus a single dose of 400 mg of albendazole or 10 mg base/kg of pyrantel pamoate for treatment of intestinal nematodiasis including 1 864 cases infected with hookworm, 1 568 cases infected with Ascaris, 1 785 cases in...

对成人钩虫感染者1864例、蛔虫感染者1568例和鞭虫感染者1785例及儿童蛲虫感染者373例，随机分组，比较服用单剂复方阿苯达唑3片或2片与单剂阿苯达唑400mg或噻嘧啶30mg（含基质10mg）／kg的驱虫效果和副作用。

The literature about the synthesis of the ion exchange and chelating adsorbents used in the off-line separation and preconcentration of the noble metals and the development of the on-line microcolumn separation and preconcentration of the noble metals were reviewed. Four silica gel-based adsorbents with rhodanine, 2-mercaptopyrimidine, 2-mercaptothiazoline and isophenylthiourea as the functional groups were first synthesized and applied to the on-line separation and preconcentration of silver, gold, palladium and platinum for their FAAS determination.

本论文在回顾螯合吸附材料的合成及其在贵金属的离线和流动注射在线预浓集分离发展状况的基础上，首次合成了含罗丹宁、2-巯基嘧啶、2-巯基噻唑啉和异二苯基硫脲等四种以硅胶为载体的螯合吸附剂，并用于银、金、钯和铂的流动注射微填充柱在线预浓集分离、火焰原子吸收光谱分析。

VITEK GNS-506 was used to detect ESBLs, and was compared with double-disk synergy test. Results Among 48 strains of K.pneumoniase detected using VITEK GNS-506, 24 strains were found to be ESBLs positive, and 24 strains ESBLs negative.

用VITEK-AMS专用药敏卡GNS-506进行ESBLs检测，并以头孢曲松、头孢噻肟、头孢他啶和氨曲南为底物，用纸片协同试验作对照。

The determination of high molecular weight impurities which existed in cefotaxime, ceftriaxone and ceftazidime and the influences of different ion-pair reagents; pH value of the eluants and the flow rate on the chromatographic column were discussed in detail.

以建立头孢噻肟、头孢曲松、头孢他啶中高分子杂质含量的快速测定方法为目的，对不同离子对试剂、洗脱剂pH、洗脱剂类型、离子对浓度、洗脱速度等因素进行了研究。

Three standard and two isolated strains of E.coli were used for drug sensitivity test on Chloramphenicol, Ciprofloxacin Lactate, Rifampicin, sulfamonomethoxine, Florfenicol, Ceftiofur Sodium as well as the antimicrobial synergists sulbactam sodium and TMP. The bacteriostasis results of the antibiotics against E.coli In vitro were compared when they were used separately or combined with the synergist.

试验用3株大肠杆菌标准株和2株地方分离株，选择氯霉素、乳酸环丙沙星、利福平、磺胺-6-甲氧嘧啶钠、氟苯尼考、头孢噻呋和抗菌增效剂舒巴坦钠、TMP进行药敏试验，比较几种药物单一或与增效剂合用对大肠杆菌的体外抑菌效果。

AIM: To investigate the platelet aggregations in patients with coronary heart disease and the effect of ticlopidine treatment.

目的：探讨冠心病患者血小板聚集功能以及噻氯匹啶对此过程的抑制作用。

He and Nina moved to California and lived at 2005 Ivar Street, Apt.

他和Nina搬到加州，并在2005年伊瓦尔街，公寓生活。

Droperidol （ potently inhibits transfected HERGchannels and this is the probable mechanism for QT prolongation.

氟哌利多有效地抑制了转染的 HERG 钾通道，可能是 QT 间期延长的机制。