查询词典 activity

In this paper, the stable Au complexes are classified according to the coordination atoms and their characteristic structure. The recent development of the researches on the antitumor activity of Au complexes including the structure-activity relationship, biological targets and the mechanisms of action are reviewed. The structure of the coordination ligand and the leaving group have great impact on the in vitro cytotoxicity of the Au complex. Many physical and biological methods are introduced to study the interaction between the Au complexes and the suspected bio-target, such as DNA, protein, mitochondrion, thio-containing biomolecules, etc. The interaction modes (intercalating, electrostatic interaction, covalent bonding, etc.) are focused to illustrate the reason for the antitumor activity of Au complexes.

本文按配位原子的不同总结了稳定三价金配合物的结构特征，按其生物活性的构效关系、生物靶点和作用机制综述了三价金配合物抗肿瘤活性研究的最新成果：配体的结构特点以及离去基团对三价金配合物的体外细胞毒性影响较大；介绍了用于检测三价金配合物与可能的生物靶分子之间的相互作用的多种物理和生物学方法，重点关注了相互作用的模式，如嵌入/静电吸引/共价结合等，并解释了三价金配合物抗肿瘤活性的原因。

In this paper, the stable Au complexes are classified according to the coordination atoms and their structural characteristics. The recent development of the researches on the antitumor activity of Au complexes including the structure-activity relationships, biological targets and the mechanisms of action are reviewed. The structure of the coordination ligand and the leaving group have great impact on the in vitro cytotoxicity of the Au complex. Many physical and biological methods are introduced to study the interaction between the Au complexe and the suspected bio-target, such as DNA, protein, mitochondrion, thio-containing biomolecules, etc. The interaction modes (intercalating, electrostatic interaction, covalent bonding, etc.) are focused to illustrate the reason for the antitumor activity of Au complexes.

本文按配位原子的不同总结了稳定三价金配合物的结构特征，按其生物活性的构效关系、生物靶点和作用机制综述了三价金配合物抗肿瘤活性研究的最新成果：配体的结构特点以及离去基团对三价金配合物的体外细胞毒性影响较大；介绍了用于检测三价金配合物与可能的生物靶分子之间相互作用的多种物理和生物学方法，重点关注了相互作用的模式，如嵌入/静电吸引/共价结合等，并解释了三价金配合物抗肿瘤活性的原因。

Practice got rid of the category of ethical and moral behavior, Practice signified "the real and perceptual activity" of people, namely people started from their own need, unceasing negatived extant world by the way of themselves, accelerated the world to turn into the real world, the activity is social and historical activity.

马克思科学实践观的确立，使&实践&摆脱伦理道德行为的范畴，&实践&指人的&现实的、感性的活动&，即从人的自身的需要出发，用自身的方式去不断地否定现存世界，促使其向&应然&世界转化的活动，是社会的活动，是历史的活动。

Based on the analysis on the oil sources and migration pathway of this area, the mineralization modes of the oil sand in the area are derived in this paper. Main conclusions are drawn as follows: a. multiphase tectonic activity resulted in multistage hydrocarbon generation of the source rock; b. threestage tectonic activity and threestage mineralization process formed a great deal of unconformity and fault pathway, thus the crude oil could migrate in a long distance; c. the tectonic activity in Yanshan and Himalayan stages uplifted the edge of the basin and the eroded reservoir outcropped to the surface, the light oil escaped and then the oil sand resource formed; d.

通过对该区油源和运移通道的分析研究，得出该区油砂的成矿模式：①多期的构造活动使烃源岩多期生烃；②三期构造活动、三个阶段的成矿过程，形成了大量的不整合面和断层通道，使原油远距离运移；③燕山期和喜马拉雅期构造活动使盆地边缘抬升，经受剥蚀，油层出露地表，轻质油逸散形成了现今的油砂资源。

85 And 119486/79. They are a novel type of antibiotic having both the wide antibacterial spectrum and high safety of penicillin and cephem antibiotics belonging to beta -lactam antibiotics, as well as the potent antibacterial activity and high beta -lactamase stability of carbapenem antibiotics.Sodium-(5R, 6S)-6-[-1-hydroxyethyl]-7-oxo-3- [-2-tetrahydrofuryl]-4-thia-1-azabicyclo [3.2.0] hept-2-ene-2-carboxylate 5/2 hydrate (faropenem sodium, hereinafter referred to as compound 1) is currently used as an oral drug for various infectious diseases and is reported to show potent antibacterial activity against not only methicillin-sensitive Staphylococcus aureus, Streptococcus pyrogenes and Streptococcus pneumoniae but also gram-positive bacteria for which conventional beta -lactam drugs have proved ineffective such as penicillin-resistant pneumococci, oral staphylococci and enterococci, also showing a wide antibacterial spectrum covering gram-negative bacteria such as Haemophilus influenzae and anaerobic bacteria such as the genus Bacteroides, which activity is due to its novel skeleton penem ring (Kagaku Ryoho no Ryoiki The Field of Chemotherapy, Vol.

他们是一种新型的抗生素都具有广泛的抗菌谱和高度的安全青霉素和cephem抗生素，属于β-内酰胺类抗生素，以及作为强大的抗菌活性和高β-内酰胺酶稳定的碳青霉烯类antibiotics.sodium -（ 5 R ， 6 S ）-6 -[ - 1 -羟乙基] - 7 -氧- 3 - [ - 2 - t etrahydrofuryl] - 4 -硫杂- 1 -氮杂双环[ 3 。2.0]庚- 2 -节能- 2 -羧酸5 / 2水合物（法罗培南钠，以下简称为化合物1 ）是目前用来作为口服药物，为各种传染病和报道，以显示强大的抗菌活性，不仅对甲氧敏感的金黄色葡萄球菌，链球菌pyrogenes和肺炎链球菌，但也克阳性菌为常规β-内酰胺类药物已证明无效，如青霉素耐药pneumococci ，口腔葡萄球菌和肠球菌，也显示出广泛的抗菌谱，包括革兰阴性菌如流感嗜血杆菌和厌氧菌如属杆菌，这活动是由于其新颖的骨架青霉烯环（（化学ryoho没有ryoiki领域的化疗），第13卷，第10号，第74-80 ， 1997年）。

The maximum activity appeared at 96h PI(23.70±7.65);in the dose-effective ness experiment,40 broilers were inoculated with different doses of sporulated oocysts respectively:there were 0,0.5×104,1.0×104,1.5×104,2.0×104, 2.5×104,3.0×104,3.5×104per chicken,iNOS activity was examined by the same method at the time with maximum iNOS activity detected in the experiment of time-effective relationship after PI.

试验结果表明，与对照组相比，肉鸡盲肠组织iNOS的活性在接种球虫后不同时间明显不同，其中接种后第96h活性最高(23.70±7.65)；在剂量－效应关系试验中，40只肉鸡以不同的剂量0、0.5×104、1.0×104、1.5×104、2.0×104、2.5×104、3.0×104、3.5×104个/只分别口服接种，然后按时间－效应关系中酶活性最高的时间点取样，以同法检测iNOS活性。

The supported WP catalysts showed considerable activity in HDS reaction of dibenzothiophene and HDN reaction of quinoline. The ibenzothiophene HDS activity and quinoline HDN activity of the spported WP catalysts synthesized by co-impregnation method was better than that synthesized by mixing method. The HDS and HDN activities of 25～30% WP catalysts synthesized by co-impregnation method and reduced at 650～750℃ were better than those of the corresponding sulfurized catalyst.

负载型WP催化剂具有较好的二苯并噻吩加氢脱硫和喹啉加氢脱氮活性，共浸渍法制备的磷化钨催化剂二苯并噻吩加氢脱硫和喹啉加氢脱氮活性要高于混合法制备的磷化钨催化剂。650～750℃还原制备的负载量25～30%的浸渍法磷化钨催化剂具有较高的二苯并噻吩加氢脱硫和喹啉加氢脱氮活性，高于相应的硫化态催化剂。

The results showed that as the leaves development, POD activity on leaves of the male sterility line significantly differed from that in the maintainer and restorer line. The CAT activity had little difference in tasseling stage, SOD activity in the male sterility line was higher than its maintainer and restorer line, and the difference was significant in every stages.

结果表明：玉米叶片在生长过程中，不育系与保持系和恢复系叶片中的POD活性有明显差异；CAT活性在抽雄期相差不大；不育系每个时期的SOD活性均显著高于保持系。

The two NS5B proteins showed the same RdRp activity changes to these three templates: they had the highest activity using 3'terminuses from HCV genotype 2a negative RNA strand as template and the lowest activity using 3'terminuses of HCV genotype 1b negative RNA strand as template.

两种NS5B蛋白对HCV 1a、1b和2a型负链3'末端RNA模板表现出相同的活性差异，两种蛋白均对2a型负链3'末端RNA模板表现出最高的聚合酶活性，对1b型负链3'末端RNA模板表现出最低的酶活性。

This article starts from the activity theory, It has analyzed the activity characteristics, including task activity, motion , operation, as well as the dynamic relations between them .

本文从活动理论入手，详细分析了任务型学习的活动特征，包括任务活动、行动、语言操作，以及它们之间的动态关系。

In the chapter 2, the theoretic knowledge about the photosensitive resin and the grinding tools was firstly introduced.

第二章阐述了光固化树脂结合剂磨具的相关理论研究。

Do not use the program's indenting or margin-setting features; these will be added during typesetting.

不要使用缩排，页面边缘设置之类的选项，偶看不大懂。